Pimozide-d4 is a deuterium labeled Pimozide. It acts as a dopamine receptor antagonist with Ki values of 1.4 nM, 2.5 nM, and 588 nM for dopamine D2, D3, and D1 receptors, respectively. It also has an affinity at α1-adrenoceptor with a Ki of 39 nM, and inhibits STAT3 and STAT5. This compound can be used as a tracer or as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
- Deuterium labeled compound
- Dopamine receptor antagonist (D2, D3, D1)
- Affinity at α1-adrenoceptor
- Inhibits STAT3 and STAT5
- Can be used as a tracer
- Can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS